Microwave-Induced Synthesis of Aromatic Heterocycles
Microwave-Induced Synthesis of Aromatic Heterocycles

Author: Abdul Rauf

Publisher: Springer Science & Business Media

Published: 2011-09-18

Total Pages: 98

ISBN-13: 9400714858

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For more than a century, heterocycles have played a crucial role in the biological and industrial development of society, becoming one of the most researched areas within organic chemistry. The first chapter of Microwave-Induced Synthesis of Aromatic Heterocycles is based on microwave theory, the latest developments in instrumentation technology, and the various microwave technologies used for synthesis. The remainder of the chapters are divided into two sections. Section A deals with the five-membered heterocycles (pyrazoles, isoxazoles, triazoles, oxadiazoles, thiazoles, imidazoles, oxazoles, oxazolines etc.) and in Section B, various six-membered heterocycles (triazines, benzoxazoles, benzimidazoles, benzothiazoles) are presented. Both sections contain a detailed, recent literature review of microwave assisted synthesis and its applicability to various aromatic heterocyclics.

Microwave Assisted Organic Synthesis
Microwave Assisted Organic Synthesis

Author: Jason Tierney

Publisher: John Wiley & Sons

Published: 2009-02-12

Total Pages: 296

ISBN-13: 1405168447

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The first reports on the application of microwaves in organicsynthesis date back to 1986, but it was not until the recentintroduction of specifically designed and constructed equipment,which countered the safety and reproducibility concerns, thatsynthetic application of microwaves has become established as alaboratory technique. Microwave assisted synthesis is now beingadopted in many industrial and academic laboratories to takeadvantage of the novel chemistry that can be carried out using avariety of organic reaction types. This book demonstrates the underlying principles of microwavedielectric heating and, by reference to a range of organic reactiontypes, it's effective use in synthetic organic chemistry. Toillustrate the impact microwave assisted organic synthesis can haveon chemical research, case studies drawn mainly from thepharmaceutical industry are presented.

Green Synthetic Approaches for Biologically Relevant Heterocycles
Green Synthetic Approaches for Biologically Relevant Heterocycles

Author: Goutam Brahmachari

Publisher: Elsevier

Published: 2021-03-20

Total Pages: 644

ISBN-13: 0323851304

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Green Synthetic Approaches for Biologically Relevant Heterocycles, Second Edition, Volume One: Advanced Synthetic Techniques reviews this significant group of organic compounds within the context of sustainable methods and processes, expanding on the first edition with fully updated coverage and a whole range of new chapters. Volume One explores advanced synthetic techniques, with each chapter presenting in-depth coverage of various green protocols for the synthesis of a wide variety of bioactive heterocycles that are classified on the basis of ring-size and/or the presence of heteroatoms. Techniques covered range from high pressure cycloaddition reactions and microwave irradiation to sustainable one-pot domino reactions. This updated edition is an essential resource on sustainable approaches for academic researchers, R&D professionals, and students working across medicinal, organic, natural product and green chemistry. - Provides fully updated coverage of the field of greener heterocycle synthesis - Includes new chapters on varied multicomponent reactions, alongside both traditional and novel approaches - Presents information in an accessible style with an emphasis on sustainability

Bioactive Peptides
Bioactive Peptides

Author: John Onuh

Publisher: CRC Press

Published: 2021-06-14

Total Pages: 527

ISBN-13: 1000387550

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Bioactive peptides have been receiving attention recently due to their applications as health-promoting agents. Derived from food proteins and other natural sources, they exhibit various beneficial effects such as preventing diseases or modulating physiological systems once absorbed. As the market for nutraceuticals and functional foods continues to expand, consumer interest has also grown and there are many common foods that have shown an abundance of bioactive peptides, including dairy products, cereal, legumes, meat, and numerous other sources. In this newest addition to the series Nutraceuticals: Basic Research and Clinical Applications, Bioactive Peptides: Production, Bioavailability, Health Potential, and Regulatory Issues provides a comprehensive review of the current state of knowledge in the field of food protein hydrolysates and bioactive peptides, their food sources, bioavailability, production, applications, functionalities, health potentials, and regulatory issues governing their use. Features Discusses different methodologies employed for scaling up bioactive peptides commercially Provides information on optimizing the production process Explains various bioactive properties exerted by different types of bioactive peptides Explores the application of metabolomics to the study of bioactive peptides With over 20 chapters written by established subject matter experts in their field, this book provides timely information and discusses the latest developments of bioactive peptides. It will be useful for researchers, academics, and industry experts, and can serve as an excellent resource for anyone interested in enhancing their knowledge in the field of bioactive peptides.

Chemical Drug Design
Chemical Drug Design

Author: Girish Kumar Gupta

Publisher: Walter de Gruyter GmbH & Co KG

Published: 2016-10-10

Total Pages: 298

ISBN-13: 311036882X

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Chemical Drug Design provides a compact overview on recent advances in this rapidly developing field. With contributions on in silico drug design, natural product based compounds, as well as on ligand- and structure-based approaches, the authors present innovative methods and techniques for identifying and synthetically designing novel drugs.

Green Synthetic Approaches for Biologically Relevant Heterocycles
Green Synthetic Approaches for Biologically Relevant Heterocycles

Author: Goutam Brahmachari

Publisher: Elsevier

Published: 2021-02-26

Total Pages: 642

ISBN-13: 0128205865

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Green Synthetic Approaches for Biologically Relevant Heterocycles, Second Edition, Volume One: Advanced Synthetic Techniques reviews this significant group of organic compounds within the context of sustainable methods and processes, expanding on the first edition with fully updated coverage and a whole range of new chapters. Volume One explores advanced synthetic techniques, with each chapter presenting in-depth coverage of various green protocols for the synthesis of a wide variety of bioactive heterocycles that are classified on the basis of ring-size and/or the presence of heteroatoms. Techniques covered range from high pressure cycloaddition reactions and microwave irradiation to sustainable one-pot domino reactions. This updated edition is an essential resource on sustainable approaches for academic researchers, R&D professionals, and students working across medicinal, organic, natural product and green chemistry. Provides fully updated coverage of the field of greener heterocycle synthesis Includes new chapters on varied multicomponent reactions, alongside both traditional and novel approaches Presents information in an accessible style with an emphasis on sustainability

Chemistry and Biology of Beta-Lactams
Chemistry and Biology of Beta-Lactams

Author: Bimal Krishna Banik

Publisher: CRC Press

Published: 2024-11-07

Total Pages: 474

ISBN-13: 1040146627

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Due to their medicinal activity and potential use as synthetic starting materials, studies on beta-lactams have increased significantly. This unique volume takes readers on a tour de force from the concept of antibiosis to the serendipity of antibiotics, evolution of beta‐lactam development, and molecular biology of antibiotic resistance. These areas of research have culminated in a deeper understanding of microbiology, particularly in the area of bacterial cell wall synthesis and recycling. Considerable work has been performed by chemists and biologists to continue updating their findings about beta-lactam synthesis. Features: • Stereoselective synthesis of monocyclic, bicyclic, and polycyclic beta-lactams • Microwave, ultrasound, and solid support-mediated preparation of beta-lactams • Diverse medicinal activities including anticancer activities of beta-lactams and products obtained from them • Nanoparticles, artificial intelligence, and dipole moments in beta-lactam science • Synthesis and mechanism of formation of polyaromatic beta-lactams

Green Chemistry: Synthesis of Bioactive Heterocycles
Green Chemistry: Synthesis of Bioactive Heterocycles

Author: K. L. Ameta

Publisher: Springer

Published: 2014-06-17

Total Pages: 418

ISBN-13: 8132218507

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The book presents a succinct summary of methods for the synthesis and biological activities of various different-sized bioactive heterocycles using different green chemistry synthetic methodologies, like microwave, ultrasonic, water mediated, ionic liquids, etc. The book also provides an insight of how green chemistry techniques are specific to the bioactive heterocyclic compounds.

Iodine-Assisted Synthesis of Six- and Seven-Membered Heterocycles
Iodine-Assisted Synthesis of Six- and Seven-Membered Heterocycles

Author: Navjeet Kaur

Publisher: Elsevier

Published: 2023-02-09

Total Pages: 382

ISBN-13: 0443152268

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Iodine-Assisted Synthesis of Six- and Seven-Membered Heterocycles covers both existing and the latest methods for the synthesis of various six- and seven-membered heterocycles using iodine. Covering an important and rapidly growing branch of heterocyclic chemistry, this book allows users easy access to the synthetic protocols for the synthesis of heterocycles, acting as a guide for how to make these important compounds employed as agrochemicals, pharmaceuticals, and veterinary products, using particular reagents. This book will be of interest to students, pharmacologists, biochemists, and organic and medicinal chemists. - Covers different methodologies for the synthesis of six- and seven-membered heterocycles using iodine - Includes the applications of six- and seven-membered heterocycles - Includes reactions schemes, mechanisms, and illustrations of the structure of reactive intermediates

Advances in Microwave Chemistry
Advances in Microwave Chemistry

Author: Bimal K Banik

Publisher: CRC Press

Published: 2018-12-07

Total Pages: 415

ISBN-13: 1351240471

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Advances in Microwave Chemistry discusses the novel bond formation methodologies, synergistic effects of microwaves with other entities, sample preparation including digestion, combustion, and extraction techniques, as well as selectivity in chemical processes. Recent updates are provided on microwave-assisted syntheses of pharmacologically significant aza-, oxo- and other heterocycles, including lactams, nucleosides, bile acids and sterols, the preparation of nanomaterials, composites, and absorber layer materials for thin film. This book also incorporates comparative discussions involving microwave irradiation with conventional methods in different aspects of organic, inorganic, medicinal, and green chemistry. Key Features: Provides a comparative discussion on microwave irradiation with conventional methods in different aspects of organic, inorganic, medicinal, and green chemistry Presents recent applications of microwave radiation in biocatalysis Offers a complete package correlating various aspects of microwaves in organic syntheses, the biological impact of products formed in reactions, pharmacological features, and environmental sustainability of the procedures Explains microwave-induced reactions on structurally complex bile acids and sterols Stands as a valuable and unique addition to the well-established book series, New Directions in Organic and Biological Chemistry